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        RG2833, ≥98%
        ??【編號(hào)】:127721

        ??【產(chǎn)品名稱】:RG2833, ≥98%

        ??【規(guī)格】:5MG

        ??【用途】:

          RG2833, ≥98%

          Product Name: RG2833
          CAS號(hào):1215493-56-3
          分子式:C20H25N3O2
          分子量:339.43
          貯存: 儲(chǔ)存溫度-20°C
          可溶性: 25°C: DMSO
          生化和生理學(xué)機(jī)理:
          Description:
          IC50 Value: N/A
          RGFP 109 is a histone deacetylase inhibitor which can attenuate L-DOPA-induced dyskinesia in the MPTP-lesioned marmoset.
          in vitro: N/A
          in vivo: RGFP109 had no acute effects on dyskinesia after single or 6 days once-daily treatment (both P > 0.05). However, one week following cessation of RGFP109, dyskinesia and duration of ON-time with disabling dyskinesia were reduced by 37% and 50%, respectively (both P < 0.05), compared to that seen previously with L-DOPA alone. There was no change in anti-parkinsonian actions of, or ON-time duration afforded by, L-DOPA (P > 0.05) [1].
          Clinical trial: Phase 1
        上一篇:利福昔明,≥99% 下一篇:Retaspimycin



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